SCHEMBL8896293

SCHEMBL8896293

COC(=O)CCc1ccc(N2CCN(C3CCC4CN(C)CCC4C3)C2=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.40
EPHX2 P34913 1/20 0.36
S1PR1 P21453 1/20 0.35
F10 P00742 3/20 0.35
HPN P05981 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
HGFAC Q04756 1/20 0.35
ST14 Q9Y5Y6 1/20 0.35
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
TP53 P04637 1/20 0.33
F2 P00734 1/20 0.33
HDAC1 Q13547 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8897736 0.84 KHK (0.37) HRH3EPHX2S1PR1F10HPN
SCHEMBL8985758 0.81 HRH3 (0.39) HRH3EPHX2ALDH1A1CYP3A4
SCHEMBL8895805 0.81 HRH3 (0.39) HRH3EPHX2ALDH1A1CYP3A4
SCHEMBL7282065 0.81 HRH3 (0.41) HRH3EPHX2S1PR1F10HPN
SCHEMBL7273643 0.80 HRH3 (0.43) HRH3EPHX2S1PR1F10HPN
Hydrochloric Acid SCHEMBL7394184 0.80 HRH3 (0.41) HRH3EPHX2S1PR1F10HPN
SCHEMBL7280320 0.78 KHK (0.48) HRH3EPHX2S1PR1F10ALDH1A1
SCHEMBL7272988 0.77 F10 (0.54) F10HPNPRSS1PRSS2PRSS3
SCHEMBL7282879 0.77 F10 (0.46) HRH3S1PR1F10HPNPRSS1
SCHEMBL8575577 0.75 HRH3 (0.42) HRH3EPHX2S1PR1F10HPN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed