SCHEMBL8897551

SCHEMBL8897551

CCCC(=O)NS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)cc2-c2ccccc2Cl)cc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.63
PTGS1 P23219 7/20 0.63
HDAC3 O15379 4/20 0.51
HDAC1 Q13547 4/20 0.51
HDAC2 Q92769 4/20 0.51
HDAC8 Q9BY41 4/20 0.51
HDAC6 Q9UBN7 4/20 0.51
HDAC4 P56524 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
PDPK1 O15530 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904051 0.88 PTGS2 (0.69) PTGS2PTGS1PDPK1
SCHEMBL5073550 0.85 PTGS2 (0.61) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL15422948 0.82 HDAC3 (0.71) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL3244766 0.78 PTGS2 (1.00) PTGS2PTGS1PDPK1
SCHEMBL5069836 0.77 PTGS2 (0.64) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL5858032 0.75 PTGS2 (0.70) PTGS2PTGS1PDPK1
SCHEMBL3114291 0.74 HDAC3 (0.73) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL27811209 0.74 HDAC3 (0.51) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL27789922 0.74 HDAC3 (0.47) PTGS2PTGS1HDAC3HDAC1HDAC2
SCHEMBL6251010 0.74 HDAC3 (0.68) PTGS2PTGS1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO claimed