SCHEMBL8897713

SCHEMBL8897713

CCOC(=O)C(C)Cc1ccc(NC(=O)N(CC(OCC)OCC)c2ccc3c(c2)CCN(C(=O)C(F)(F)F)CC3)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
ATM Q13315 1/20 0.34
GAA P10253 1/20 0.34
EPHX2 P34913 1/20 0.33
PPARG P37231 1/20 0.33
TNF P01375 2/20 0.33
NOD1 Q9Y239 2/20 0.33
NOD2 Q9HC29 1/20 0.33
NPY1R P25929 1/20 0.33
NPY2R P49146 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8897664 0.84 KMT2A (0.37) MEN1KMT2AESR1ESR2NPC1
SCHEMBL8897546 0.74 ESR1 (0.38) ESR1ESR2
SCHEMBL8897540 0.74 ESR1 (0.38) ESR1ESR2
SCHEMBL8895079 0.74 ESR1 (0.39) MEN1KMT2AESR1ESR2RAB9A
SCHEMBL8895074 0.74 ESR1 (0.39) MEN1KMT2AESR1ESR2RAB9A
SCHEMBL8562345 0.73 ESR1 (0.39) ESR1ESR2NPC1RAB9AEPHX2
SCHEMBL8896472 0.73 ESR1 (0.35) ESR1ESR2
SCHEMBL8559726 0.71 ESR1 (0.46) MEN1KMT2AESR1ESR2NPC1
SCHEMBL8562326 0.71 ESR1 (0.33) ESR1ESR2KDM4EALDH1A1
SCHEMBL8558150 0.71 ESR1 (0.35) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed