SCHEMBL8559726

SCHEMBL8559726

CCOC(CNc1ccc2c(c1)CCN(C(=O)C(F)(F)F)CC2)OCC

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.46
ESR2 Q92731 3/20 0.46
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ABHD6 Q9BV23 4/20 0.38
KDM4E B2RXH2 1/20 0.37
TYRO3 Q06418 2/20 0.36
MERTK Q12866 2/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471562 0.89 ESR1 (0.50) ESR1ESR2HDAC6ABHD6KDM4E
SCHEMBL7363844 0.78 NAMPT (0.43) POLBNPC1RAB9AEPHX1EPHX2
SCHEMBL7418167 0.76 ESR1 (0.46) ESR1ESR2MEN1KMT2AHDAC6
SCHEMBL719483 0.75 ESR1 (0.52) ESR1ESR2HDAC6NPC1RAB9A
SCHEMBL7424343 0.74 MAPT (0.51) NPC1RAB9A
SCHEMBL7422272 0.74 ESR1 (0.51) ESR1ESR2HDAC6ABHD6KDM4E
SCHEMBL8562609 0.72 ESR1 (0.44) ESR1ESR2NPC1RAB9A
SCHEMBL7422278 0.70 ALDH1A1 (0.54)
SCHEMBL2309023 0.70 ESR1 (0.85) ESR1ESR2HDAC6ABHD6
SCHEMBL13334504 0.69 ESR1 (0.56) ESR1ESR2MEN1KMT2AABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed