SCHEMBL8898972

SCHEMBL8898972

CS(=O)(=O)c1cccc(C(N)(CO)C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.49
GRM2 Q14416 2/20 0.44
GRM3 Q14832 2/20 0.44
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
HSD17B10 Q99714 1/20 0.41
LOXL2 Q9Y4K0 3/20 0.39
LOX P28300 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
CYP2D6 P10635 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
DRD2 P14416 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30628251 0.75 KIF11 (0.47) KIF11GRM2GRM3ALDH1A1GAA
SCHEMBL28838841 0.75 KIF11 (0.47) KIF11GRM2GRM3CYP1A2CYP2C19
SCHEMBL17420495 0.75 KIF11 (0.47) KIF11GRM2GRM3ALDH1A1GAA
SCHEMBL1712451 0.75 CYP1A2 (0.47) KIF11ALDH1A1CYP1A2CYP2C19CYP2D6
SCHEMBL1712450 0.75 CYP1A2 (0.47) KIF11ALDH1A1CYP1A2CYP2C19CYP2D6
SCHEMBL1712531 0.75 CYP1A2 (0.47) KIF11ALDH1A1CYP1A2CYP2C19CYP2D6
SCHEMBL4631894 0.74 KIF11 (0.51) KIF11GRM2GRM3LOXL2LOX
Hydrochloric Acid SCHEMBL8064648 0.73 CYP1A2 (0.46) KIF11ALDH1A1CYP1A2CYP2C19CYP2D6
SCHEMBL30087634 0.71 KIF11 (0.46) KIF11SMN1; SMN2NPSR1
SCHEMBL12157465 0.71 KIF11 (0.48) KIF11ALDH1A1GAAHSD17B10CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507153-B1 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORP (US) 1997-07-09 EP claimed
US-5346828-A Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase CELGENE CORPORATION (US) 1994-09-13 US claimed
EP-0507153-A2 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORPORATION (US) 1992-10-07 EP claimed