Bromide

Bromide

SCHEMBL8900274

CC(C)(C)OC(=O)Oc1cccc(CN2CC[C@@H]([P+](c3ccccc3)(c3ccccc3)c3ccccc3)C2=O)c1.[Br-]

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP7 P09237 1/20 0.38
MMP10 P09238 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
MMP14 P50281 1/20 0.38
ADAM17 P78536 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CCR8 P51685 3/20 0.36
KDM4E B2RXH2 1/20 0.35
NPY1R P25929 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8560227 1.00 APP (0.38) APPMMP1MMP2MMP7MMP10
Bromide SCHEMBL8563260 0.83 SIGMAR1 (0.50) KMT2AMEN1KDM4E
Bromide SCHEMBL8901003 0.83 SIGMAR1 (0.50) KMT2AMEN1KDM4E
Bromide SCHEMBL8898969 0.83 KMT2A (0.38) MMP1MMP2MMP9ADAM17KMT2A
Bromide SCHEMBL8567797 0.83 KMT2A (0.38) MMP1MMP2MMP9ADAM17KMT2A
Bromide SCHEMBL8565335 0.80 SIRT2 (0.48) KMT2AMEN1
Bromide SCHEMBL8562348 0.78 SCN1A (0.35) KDM4E
Bromide SCHEMBL8563395 0.77 HDAC1 (0.43) KMT2AMEN1
Bromide SCHEMBL8563399 0.77 HDAC1 (0.43) KMT2AMEN1
Bromide SCHEMBL7619358 0.77 PLA2G10 (0.45) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed