SCHEMBL8900403

SCHEMBL8900403

CCCN1CCC2c3cccc(OC)c3CCC21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 19/20 1.00
DRD2 P14416 8/20 0.71
DRD1 P21728 1/20 0.68
DRD4 P21917 1/20 0.68
DRD5 P21918 1/20 0.68
DRD3 P35462 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900398 1.00 HTR1A (1.00) HTR1ADRD2DRD1DRD4DRD5
Hydrochloric Acid SCHEMBL8900389 0.99 HTR1A (0.98) HTR1ADRD2DRD1DRD4DRD5
Hydrochloric Acid SCHEMBL8900392 0.99 HTR1A (0.98) HTR1ADRD2DRD1DRD4DRD5
SCHEMBL9119857 0.87 HTR1A (0.77) HTR1ADRD2DRD1DRD4DRD5
SCHEMBL9119868 0.87 HTR1A (0.77) HTR1ADRD2DRD1DRD4DRD5
SCHEMBL9121023 0.87 HTR1A (0.77) HTR1ADRD2DRD3
SCHEMBL9121014 0.87 HTR1A (0.77) HTR1ADRD2DRD3
SCHEMBL9119963 0.86 HTR1A (0.75) HTR1ADRD2DRD1DRD4DRD5
SCHEMBL9119950 0.86 HTR1A (0.75) HTR1ADRD2DRD1DRD4DRD5
Hydrochloric Acid SCHEMBL9441342 0.85 HTR1A (0.73) HTR1ADRD2DRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482084-B1 (1,2N) AND (3,2N)-CARBOCYCLIC-2-AMINO TETRALIN DERIVATIVES UPJOHN CO (US) 1997-05-07 EP claimed
EP-0548664-B1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives HOFFMANN LA ROCHE (CH) 1995-05-31 EP disclosed
US-5318966-A Administering the enzyme inhibitor for treating alzheimer's disease, learning enhancement, brain disorders HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
US-5318967-A Cognition activators for alzheimer's disease, learning enhancement HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
EP-0548664-A1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed