SCHEMBL8901972

SCHEMBL8901972

COc1cc(OC)c(S(N)(=O)=O)cc1C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.63
NPSR1 Q6W5P4 1/20 0.63
PKM P14618 2/20 0.59
CA12 O43570 2/20 0.54
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
CA3 P07451 2/20 0.54
CA4 P22748 2/20 0.54
CA6 P23280 2/20 0.54
CA5A P35218 2/20 0.54
CA7 P43166 2/20 0.54
CA9 Q16790 2/20 0.54
CA13 Q8N1Q1 2/20 0.54
CA14 Q9ULX7 2/20 0.54
CA5B Q9Y2D0 2/20 0.54
LCK P06239 1/20 0.51
FYN P06241 1/20 0.51
ALDH1A1 P00352 5/20 0.49
HPGD P15428 2/20 0.49
CISD1 Q9NZ45 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8573435 0.88 CA12 (0.67) KDM4ENPSR1PKMCA12CA1
SCHEMBL11158120 0.87 PKM (0.53) KDM4ENPSR1PKMCA12CA1
SCHEMBL10721933 0.87 PKM (0.56) KDM4ENPSR1PKMCA12CA1
SCHEMBL28899597 0.85 CISD1 (0.66) KDM4ENPSR1PKMCA12CA1
SCHEMBL7797968 0.84 KDM4E (0.65) KDM4ENPSR1PKMCA12CA1
SCHEMBL7801303 0.83 KDM4E (0.63) KDM4ENPSR1PKMCA12CA1
SCHEMBL10723753 0.81 KDM4E (0.61) KDM4ENPSR1PKMLCKFYN
SCHEMBL11688578 0.81 PKM (0.70) KDM4EPKMCA12CA1CA2
SCHEMBL11710380 0.81 PKM (0.50) KDM4ENPSR1PKMCA12CA1
SCHEMBL11159006 0.80 KDM4E (0.60) KDM4ENPSR1PKMLCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686482-A DOPAMINE RECEPTOR ANTAGONIST YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-11 US disclosed
EP-0757985-A1 N-(3-PYRROLIDINYL)BENZAMIDE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-02-12 EP disclosed
EP-0068700-A1 Azobicycloalkylbenzamides, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1983-01-05 EP disclosed