SCHEMBL8905959

SCHEMBL8905959

CCOC(=O)[C@@H](C[C@H](COCc1ccccc1)C(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.59
CTSS P25774 5/20 0.56
PPARG P37231 2/20 0.54
KLK7 P49862 2/20 0.50
KLK5 Q9Y337 2/20 0.50
SYK P43405 1/20 0.46
CTSK P43235 6/20 0.45
REN P00797 1/20 0.45
RAB9A P51151 1/20 0.45
CTSL P07711 2/20 0.44
CTSB P07858 1/20 0.44
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
CDC25B P30305 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5349842 1.00 PPARA (0.59) PPARACTSSPPARGKLK7KLK5
SCHEMBL8906370 1.00 PPARA (0.59) PPARACTSSPPARGKLK7KLK5
SCHEMBL6042808 0.92 PPARA (0.61) PPARACTSSPPARGKLK7KLK5
SCHEMBL6043892 0.92 PPARA (0.61) PPARACTSSPPARGKLK7KLK5
SCHEMBL5710546 0.92 PPARA (0.61) PPARACTSSPPARGKLK7KLK5
SCHEMBL3783761 0.89 PPARA (0.70) PPARACTSSPPARGKLK7KLK5
SCHEMBL27910918 0.83 PPARA (0.52) PPARACTSSPPARGSYKCTSK
SCHEMBL27675050 0.82 PPARA (0.56) PPARACTSSPPARGKLK7KLK5
SCHEMBL12053946 0.82 PPARA (0.56) PPARACTSSPPARGKLK7KLK5
SCHEMBL7518373 0.81 PPARA (0.74) PPARACTSSPPARGKLK7KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5659065-A CHEMICAL INTERMEDIATES FOR MEDICINAL ACTIVE AGENTS NOVARTIS CORPORATION (US) 1997-08-19 US disclosed
EP-0678500-A1 Alpha-amino alkanoic acids and reduction products as intermediates in the preparation of renin inhibitors CIBA-GEIGY AG (CH) 1995-10-25 EP disclosed