SCHEMBL8906012

SCHEMBL8906012

CCCCc1nc2ccc(C(=O)O)cc2[nH]1

nearest known ligand 0.71

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.71
ALDH1A1 P00352 2/20 0.67
MAPK1 P28482 1/20 0.67
NPSR1 Q6W5P4 1/20 0.66
HSP90AA1 P07900 1/20 0.58
ESR2 Q92731 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
TOP2A P11388 1/20 0.57
MPL P40238 1/20 0.57
KMT2A Q03164 1/20 0.52
MAPT P10636 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5387954 0.95 APEX1 (0.67) APEX1ALDH1A1MAPK1NPSR1HSP90AA1
SCHEMBL7334282 0.95 APEX1 (0.67) APEX1ALDH1A1MAPK1NPSR1HSP90AA1
SCHEMBL3639896 0.92 APEX1 (0.74) APEX1ALDH1A1MAPK1NPSR1HSP90AA1
SCHEMBL8788713 0.89 APEX1 (0.56) APEX1ALDH1A1MAPK1NPSR1TOP2A
SCHEMBL5396738 0.85 NPSR1 (0.73) APEX1ALDH1A1MAPK1NPSR1HSP90AA1
SCHEMBL8632170 0.85 MAPT (0.64) APEX1ALDH1A1MAPK1NPSR1KMT2A
SCHEMBL18229547 0.85 HDAC6 (0.68) APEX1ALDH1A1MAPK1MAPTHDAC6
Guanidine SCHEMBL8688512 0.84 APEX1 (0.55) APEX1ALDH1A1MAPK1NPSR1TOP2A
SCHEMBL7334277 0.84 APEX1 (0.53) APEX1ALDH1A1MAPK1NPSR1
SCHEMBL11376990 0.84 PARP1 (0.63) APEX1ALDH1A1MAPK1NPSR1MPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed
US-5587393-A ANGIOTENSIN ANTAGONIST USEFUL IN TREATING HYPERTENSION DR. KARL THOMAE GMBH (DE) 1996-12-24 US disclosed
US-5385925-A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1995-01-31 US disclosed