SCHEMBL8906210

SCHEMBL8906210

COc1cc([O])c(Cc2ccc3c(Cl)cccc3c2)c(O)c1C=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.41
ERN1 O75460 3/20 0.35
PDE10A Q9Y233 5/20 0.35
AR P10275 1/20 0.34
PTGES O14684 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33
TUBB8 Q3ZCM7 1/20 0.33
TUBA3E Q6PEY2 1/20 0.33
TUBA1A Q71U36 1/20 0.33
TUBA1C Q9BQE3 1/20 0.33
TUBB6 Q9BUF5 1/20 0.33
TUBB2B Q9BVA1 1/20 0.33
TUBB1 Q9H4B7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8906218 0.91 CETP (0.44) CETPERN1PDE10AAR
SCHEMBL8905392 0.86 NQO1 (0.36) ERN1ARCASP1CASP7
SCHEMBL8734491 0.84 CETP (0.39) CETPPDE10A
SCHEMBL8904879 0.79 AR (0.37) ERN1ARCASP1CASP7
SCHEMBL8732768 0.78 AR (0.40) AR
SCHEMBL8905400 0.78 NQO1 (0.37) CETPERN1ARCYP1A2CYP3A4
SCHEMBL8904212 0.78 ERN1 (0.36) ERN1CYP1A2
SCHEMBL8904950 0.76 ERN1 (0.38) ERN1
SCHEMBL8736522 0.75 THRA (0.40)
SCHEMBL8904858 0.75 ERN1 (0.38) CETPERN1PDE10ATUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677342-A ANTIDIABETIC AGENT AMERICAN HOME PRODUCTS CORPORATION (US) 1997-10-14 US claimed
US-5677342-A ANTIDIABETIC AGENT AMERICAN HOME PRODUCTS CORPORATION (US) 1997-10-14 US disclosed