SCHEMBL8906392

SCHEMBL8906392

CC(C)c1ccc(S(=O)(=O)NC(=O)C(Cc2ccc(C(F)(F)F)cc2)c2ccc3c(c2)OCO3)cc1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 9/20 0.52
EDNRA P25101 9/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8952113 0.91 EDNRA (0.50) EDNRBEDNRA
Trifluoroacetic Acid SCHEMBL8908256 0.89 EDNRA (0.52) EDNRBEDNRA
SCHEMBL9263398 0.89 EDNRB (0.57) EDNRBEDNRA
Potassium SCHEMBL9263403 0.89 EDNRB (0.57) EDNRBEDNRA
SCHEMBL9267320 0.88 EDNRB (0.54) EDNRBEDNRA
Potassium SCHEMBL9267325 0.88 EDNRB (0.54) EDNRBEDNRA
SCHEMBL8906488 0.88 EDNRA (0.57) EDNRBEDNRA
SCHEMBL9272346 0.86 EDNRA (0.60) EDNRBEDNRA
Potassium Ion SCHEMBL8907336 0.86 EDNRA (0.53) EDNRBEDNRA
Potassium SCHEMBL9272349 0.86 EDNRA (0.60) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995003295-A1 ENDOTHELIN ANTAGONISTS MERCK & CO., INC. (US) 1995-02-02 WO claimed
US-5686478-A Endothelin antagonists MERCK & CO. INC. (US) 1997-11-11 US disclosed
WO-1995003295-A1 ENDOTHELIN ANTAGONISTS MERCK & CO., INC. (US) 1995-02-02 WO disclosed