SCHEMBL8906502

SCHEMBL8906502

CCCc1nc2cc(C(=O)O)ccc2n1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 5/20 0.53
HDAC6 Q9UBN7 10/20 0.50
AGTR1 P30556 1/20 0.50
AGTR2 P50052 1/20 0.50
HDAC1 Q13547 3/20 0.49
ALDH1A1 P00352 2/20 0.49
PTGER4 P35408 1/20 0.49
PKM P14618 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HSP90AA1 P07900 1/20 0.48
HSP90AB1 P08238 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
THRB P10828 1/20 0.48
PABPC1 P11940 1/20 0.48
HPGD P15428 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3643686 0.89 AGTR1 (0.53) HCAR3HDAC6AGTR1AGTR2MEN1
SCHEMBL9597035 0.89 HDAC6 (0.50) HCAR3HDAC6HDAC1ALDH1A1PTGER4
SCHEMBL9597041 0.89 HDAC6 (0.50) HCAR3HDAC6HDAC1ALDH1A1PTGER4
SCHEMBL16166414 0.85 HDAC6 (0.52) HCAR3HDAC6HDAC1ALDH1A1PTGER4
SCHEMBL17315023 0.84 HDAC6 (0.51) HCAR3HDAC6HDAC1ALDH1A1PTGER4
Hydrochloric Acid SCHEMBL20969064 0.83 HDAC6 (0.50) HCAR3HDAC6HDAC1ALDH1A1PTGER4
SCHEMBL29703917 0.83 HDAC6 (0.50) HCAR3HDAC6HDAC1ALDH1A1PKM
SCHEMBL3438310 0.82 HDAC6 (0.57) HCAR3HDAC6HDAC1PTGER4HSD17B10
SCHEMBL7069710 0.80 HPGD (0.48) HCAR3HDAC6HDAC1ALDH1A1PTGER4
SCHEMBL1726928 0.80 JAK2 (0.60) HDAC6AGTR1AGTR2HDAC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed
US-5587393-A ANGIOTENSIN ANTAGONIST USEFUL IN TREATING HYPERTENSION DR. KARL THOMAE GMBH (DE) 1996-12-24 US disclosed
US-5385925-A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1995-01-31 US disclosed