SCHEMBL8907132

SCHEMBL8907132

CCCCCCn1c(-c2ccc3nc(CCC)n(-c4ccc(-c5ccccc5)c(C(=O)O)c4C)c3c2)nc2cccnc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.40
PPARG P37231 6/20 0.38
AGTR1 P30556 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
USP2 O75604 1/20 0.38
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
CYP2C9 P11712 1/20 0.38
ACE P12821 1/20 0.38
ADRA2C P18825 1/20 0.38
TBXA2R P21731 1/20 0.38
GLRA1 P23415 1/20 0.38
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8906955 0.90 PPARG (0.42) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL8905885 0.85 TP53 (0.47) TP53PPARGAGTR1AGTR2
SCHEMBL8905751 0.85 AGTR1 (0.39) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL8905700 0.84 PPARG (0.50) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL8906713 0.82 AGTR1 (0.45) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL8905609 0.81 PPARG (0.41) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL8906316 0.81 PPARG (0.44) PPARGAGTR1KDM4EABCC3ABCC4
SCHEMBL9255379 0.81 PPARG (0.55) PPARGAGTR1AGTR2
SCHEMBL8905963 0.80 AGTR1 (0.41) PPARGAGTR1AGTR2
SCHEMBL8905974 0.80 PPARG (0.45) PPARGAGTR1KDM4EABCC3ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed