SCHEMBL8909595

SCHEMBL8909595

CC1=C(C(=O)OCc2ccccc2)N=c2cc3c(c(C)c21)=Nc1ccc(Cl)cc1-3

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.38
PTGER1 P34995 4/20 0.37
POLB P06746 1/20 0.37
ALOX5 P09917 2/20 0.36
KMT2A Q03164 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HTT P42858 1/20 0.36
GPBAR1 Q8TDU6 2/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388713 0.89 TDP1 (0.40) POLBKMT2ATDP1SLC6A2SLC6A3
SCHEMBL8909720 0.89 DHODH (0.38) DHODHPOLBKMT2ATDP1SLC6A2
SCHEMBL8909637 0.88 TDP1 (0.40) DHODHPOLBKMT2ATDP1SLC6A2
SCHEMBL8910758 0.83 DHODH (0.38) DHODHKMT2ATDP1SLC6A2SLC6A3
SCHEMBL8911173 0.81 TDP1 (0.39) POLBKMT2ATDP1SLC6A2SLC6A3
SCHEMBL8909629 0.79 CA12 (0.39) ALOX5KMT2ATDP1HTTMAPT
SCHEMBL8909809 0.76 TSHR (0.37) KMT2AMAPTL3MBTL1NPC1RAB9A
SCHEMBL8150300 0.76 MAPK1 (0.33)
SCHEMBL8910217 0.74 TDP1 (0.44) KMT2ATDP1SLC6A2SLC6A3MAPT
SCHEMBL8155106 0.74 MAOB (0.43) POLBKMT2ATDP1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed