SCHEMBL8911990

SCHEMBL8911990

CC(NC(=O)OC(C)(C)C)C1CCN(C(=O)OCc2ccccc2)C1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.52
PPARG P37231 1/20 0.52
SYK P43405 1/20 0.50
CTSL P07711 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.48
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 2/20 0.47
LCK P06239 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
PDE4B Q07343 1/20 0.45
CTSK P43235 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17494230 1.00 GPR119 (0.52) GPR119PPARGSYKCTSLSMN1; SMN2
SCHEMBL30400179 1.00 GPR119 (0.52) GPR119PPARGSYKCTSLSMN1; SMN2
SCHEMBL19195314 1.00 GPR119 (0.52) GPR119PPARGSYKCTSLSMN1; SMN2
SCHEMBL20329576 0.94 GPR119 (0.54) GPR119SYKCTSLSMN1; SMN2NPC1
SCHEMBL17946176 0.94 GPR119 (0.54) GPR119SYKCTSLSMN1; SMN2NPC1
SCHEMBL29286130 0.88 GPR119 (0.48) GPR119PPARGSYKCTSLSMN1; SMN2
SCHEMBL25245210 0.85 GPR119 (0.59) GPR119SYKSMN1; SMN2NPC1RAB9A
SCHEMBL17591749 0.85 GPR119 (0.59) GPR119SYKSMN1; SMN2NPC1RAB9A
SCHEMBL17591931 0.85 PREP (0.53) GPR119SYKCTSLMAPK1KMT2A
SCHEMBL23576031 0.85 PREP (0.53) GPR119SYKCTSLMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380874-A Pyrrolidine carbamates DAIICHI SEIYAKU CO., LTD. (JP) 1995-01-10 US claimed
JP-9143157-A None JP disclosed
JP-H09143157-A PYRROLIDINE DERIVATIVE DAI ICHI SEIYAKU CO LTD 1997-06-03 JP disclosed
US-5476950-A Aminopyrrolidine compound DAIICHI SEIYAKU CO., LTD. (JP) 1995-12-19 US disclosed
US-5416222-A Chemical intermediates to prepare pyridinocarboxylic acid derivatives with high antimicrobial activity and excellent pharmacokinetics DAIICHI SEIYAKU CO., LTD. (JP) 1995-05-16 US disclosed
US-5380874-A Pyrrolidine carbamates DAIICHI SEIYAKU CO., LTD. (JP) 1995-01-10 US disclosed
EP-0207420-B1 PYRIDONECARBOXYLIC ACID DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1992-05-06 EP disclosed
US-5098912-A Bactericides for grampositive bacteria DAIICHI SEIYAKU CO., LTD. (JP) 1992-03-24 US disclosed
EP-0207420-A2 Pyridonecarboxylic acid derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1987-01-07 EP disclosed