SCHEMBL8912700

SCHEMBL8912700

NC(C(OCc1ccccc1)OC(=O)C(=O)OC(OCc1ccccc1)C(N)C(c1ccccc1)c1ccccc1)C(c1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 6/20 0.51
SLC1A3 P43003 5/20 0.51
SLC1A2 P43004 5/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
TACR1 P25103 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.40
ALPI P09923 1/20 0.40
PKM P14618 1/20 0.40
PTGS1 P23219 1/20 0.40
XIAP P98170 1/20 0.40
SLC7A5 Q01650 1/20 0.40
SLC15A1 P46059 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912668 0.87 GLA (0.43) SLC1A1SLC1A3SLC1A2KMT2AMEN1
SCHEMBL8912527 0.87 TACR1 (0.52) SLC1A1SLC1A3SLC1A2KMT2AMEN1
SCHEMBL8916814 0.84 FFAR1 (0.44) SLC1A1SLC1A3SLC1A2KMT2AMEN1
SCHEMBL8911831 0.84 TACR1 (0.55) TACR1
SCHEMBL8911985 0.83 RAB9A (0.47) KMT2AMEN1TACR1SMN1; SMN2ALDH1A1
SCHEMBL8910978 0.82 TACR1 (0.57) TACR1
SCHEMBL8911190 0.79 TACR1 (0.55) KMT2AMEN1TACR1PPARGPPARA
SCHEMBL16430299 0.74 SLC1A3 (0.65) SLC1A1SLC1A3SLC1A2KMT2AMEN1
SCHEMBL9725774 0.73 SLC1A1 (0.68) SLC1A1SLC1A3SLC1A2KMT2AMEN1
SCHEMBL18925992 0.73 SLC1A1 (0.68) SLC1A1SLC1A3SLC1A2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629347-A TACHYKININ ANTAGONIST USED IN TREATMENT OF INFLAMMATION, MIGRAINE, POSTHERPETIC NEURALGIA MERCK SHARP & DOHME LTD. (GB) 1997-05-13 US disclosed
WO-1993001160-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO disclosed
EP-0522808-A2 Aromatic compounds, pharmaceutical compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1993-01-13 EP disclosed