SCHEMBL8914039

SCHEMBL8914039

CS(=O)(=O)OCCCCc1cccs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
ALDH1A1 P00352 5/20 0.48
TSHR P16473 3/20 0.48
KDM4E B2RXH2 1/20 0.48
USP2 O75604 1/20 0.48
LMNA P02545 1/20 0.48
MMP9 P14780 1/20 0.48
ALOX15 P16050 1/20 0.48
TAAR1 Q96RJ0 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.43
POLB P06746 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HPGD P15428 1/20 0.42
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTGS2 P35354 2/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209882 0.98 NPC1 (0.48) NPC1ALDH1A1TSHRKDM4EUSP2
SCHEMBL9217359 0.98 NPC1 (0.48) NPC1ALDH1A1TSHRKDM4EUSP2
SCHEMBL1161703 0.88 TAAR1 (0.46) NPC1ALDH1A1TSHRKDM4EUSP2
SCHEMBL628048 0.79 SMN1; SMN2 (0.51) NPC1ALDH1A1TSHRUSP2TAAR1
SCHEMBL1367928 0.78 ALDH1A1 (0.44) NPC1ALDH1A1LMNATAAR1SMN1; SMN2
SCHEMBL4490512 0.78 TAAR1 (0.53) NPC1ALDH1A1TSHRLMNATAAR1
SCHEMBL20146704 0.76 TAAR1 (0.73) NPC1ALDH1A1TSHRUSP2TAAR1
SCHEMBL21413115 0.76 TAAR1 (0.52) NPC1ALDH1A1TSHRLMNATAAR1
SCHEMBL10341120 0.74 NPC1 (0.63) NPC1ALDH1A1TSHRUSP2TAAR1
SCHEMBL6734915 0.74 TAAR1 (0.70) NPC1ALDH1A1TSHRUSP2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013060860-A1 N-ACYL-N'-PHENYLPIPERAZINE DERIVATIVES AS SRBP MODULATORS FOR USE IN THE TREATMENT OF DIABETES AND OBESITY NATIONAL UNIVERSITY OF IRELAND, MAYNOOTH (IE) 2013-05-02 WO disclosed
US-5688804-A 3-Benzylamino-2-phenyl-piperidine derivatives as substance P receptor antagonists PFIZER INC. (US) 1997-11-18 US disclosed
EP-0654029-A1 3-BENZYLAMINO-2-PHENYL-PIPERIDINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1995-05-24 EP disclosed
WO-1994003445-A1 3-BENZYLAMINO-2-PHENYL-PIPERIDINE DERIVATIVES AS SUBSTANCE P RECEPTOR ANTAGONISTS PFIZER INC. (US) 1994-02-17 WO disclosed