SCHEMBL8914485

SCHEMBL8914485

CC(=O)NCCSc1ccnc(CSc2nc3ccccc3[nH]2)c1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.52
NPC1 O15118 4/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP3A4 P08684 1/20 0.52
HTT P42858 2/20 0.46
LMNA P02545 4/20 0.46
KMT2A Q03164 3/20 0.46
HPGD P15428 1/20 0.46
CYP2E1 P05181 1/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2B6 P20813 1/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914909 0.89 POLB (0.53) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8915694 0.88 MAPT (0.49) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8915103 0.87 RAB9A (0.51) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914857 0.86 RAB9A (0.50) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8915099 0.85 NPC1 (0.53) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914814 0.85 EPHX2 (0.61) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914947 0.84 NPC1 (0.49) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8915610 0.84 NPC1 (0.52) RAB9ANPC1CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8914843 0.84 NPC1 (0.52) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914556 0.84 NPC1 (0.48) RAB9ANPC1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP claimed
US-5616581-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
US-5504082-A BACTERICIDE FOR HELICOBACTER, ANTIULCER AGENT, GASTRIC ACIDSUPPRESSOR YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-04-02 US disclosed
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP disclosed