SCHEMBL8914719

SCHEMBL8914719

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCOC(=O)c2ccccc2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.76
CYP3A4 P08684 3/20 0.76
KDM4E B2RXH2 3/20 0.76
ABCB11 O95342 3/20 0.76
TBXA2R P21731 3/20 0.76
ADRA1A P35348 3/20 0.76
SLC6A3 Q01959 3/20 0.76
ADORA3 P0DMS8 3/20 0.76
MEN1 O00255 2/20 0.76
CYP1A2 P05177 2/20 0.76
CYP2C19 P33261 2/20 0.76
KMT2A Q03164 2/20 0.76
HIF1A Q16665 2/20 0.76
HSD17B10 Q99714 2/20 0.76
ABCB1 P08183 2/20 0.76
ADRB3 P13945 2/20 0.76
OPRK1 P41145 2/20 0.76
SCN5A Q14524 2/20 0.76
TSHR P16473 2/20 0.76
NR1I2 O75469 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912955 0.89 CYP2C9 (0.60) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL8912171 0.88 KDM4E (0.74) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL9672697 0.88 KDM4E (0.68) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL9235954 0.88 CYP2C9 (0.59) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL9485314 0.88 CYP2C9 (0.81) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL7283648 0.88 CYP2C9 (0.81) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL8913291 0.88 CYP2C9 (0.81) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL11451800 0.87 KDM4E (0.83) CYP2C9CYP3A4KDM4EABCB11TBXA2R
SCHEMBL10823894 0.87 CYP2C9 (0.79) CYP2C9CYP3A4KDM4EABCB11TBXA2R
Felodipine SCHEMBL920025 0.87 CYP2C9 (1.00) CYP2C9CYP3A4KDM4EABCB11TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7196615-A None JP disclosed
US-5658934-A Aryl-substituted alkoxycarbonyl-1,4-dihydropyridine-5-carboxylic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed
JP-H07196615-A ARYL-SUBSTITUTED ALKOXYCARBONYL-1,4-DIHYDROPYRIDINE-5-CARBOXYLIC ACID ESTER BAYER AG 1995-08-01 JP disclosed