SCHEMBL8913291

SCHEMBL8913291

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCO)C1c1cccc(Cl)c1Cl

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.81
KDM4E B2RXH2 4/20 0.81
CYP3A4 P08684 4/20 0.81
ABCB11 O95342 4/20 0.81
ADORA3 P0DMS8 4/20 0.81
CYP1A2 P05177 3/20 0.81
CYP2C19 P33261 3/20 0.81
KMT2A Q03164 3/20 0.81
HIF1A Q16665 3/20 0.81
HSD17B10 Q99714 3/20 0.81
TBXA2R P21731 3/20 0.81
ADRA1A P35348 3/20 0.81
SLC6A3 Q01959 3/20 0.81
TSHR P16473 3/20 0.81
SCN5A Q14524 3/20 0.81
ALDH1A1 P00352 3/20 0.81
HPGD P15428 3/20 0.81
MAPT P10636 3/20 0.81
MEN1 O00255 2/20 0.81
ABCB1 P08183 2/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11187877 0.91 CYP2C9 (0.74) CYP2C9KDM4ECYP3A4ABCB11ADORA3
SCHEMBL7283648 0.91 CYP2C9 (0.81) CYP2C9KDM4ECYP3A4ABCB11ADORA3
SCHEMBL9485314 0.91 CYP2C9 (0.81) CYP2C9KDM4ECYP3A4ABCB11ADORA3
SCHEMBL10823894 0.90 CYP2C9 (0.79) CYP2C9KDM4ECYP3A4ABCB11ADORA3
Felodipine SCHEMBL28260282 0.90 CYP2C9 (0.95) CYP2C9KDM4ECYP3A4ABCB11ADORA3
(R)-Felodipine SCHEMBL54486 0.90 CYP2C9 (1.00) CYP2C9KDM4ECYP3A4ABCB11ADORA3
Felodipine SCHEMBL13460298 0.90 CYP2C9 (1.00) CYP2C9KDM4ECYP3A4ABCB11ADORA3
(R)-Felodipine SCHEMBL29617765 0.90 CYP2C9 (1.00) CYP2C9KDM4ECYP3A4ABCB11ADORA3
Felodipine SCHEMBL920025 0.90 CYP2C9 (1.00) CYP2C9KDM4ECYP3A4ABCB11ADORA3
Felodipine SCHEMBL26398 0.90 CYP2C9 (1.00) CYP2C9KDM4ECYP3A4ABCB11ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658934-A Aryl-substituted alkoxycarbonyl-1,4-dihydropyridine-5-carboxylic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed
EP-0371492-B1 Process for the preparation of 1,4-dihydropyridine derivatives NISSHIN FLOUR MILLING CO (JP) 1995-06-21 EP disclosed
EP-0371492-A2 Process for the preparation of 1,4-dihydropyridine derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1990-06-06 EP disclosed