SCHEMBL8914866

SCHEMBL8914866

O=C1c2ccccc2C(=O)N1CCCCCCCCCCSc1ccccc1

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.88
CYP2D6 P10635 1/20 0.88
CYP2C19 P33261 1/20 0.88
RAB9A P51151 2/20 0.76
SMN1; SMN2 Q16637 2/20 0.76
NPC1 O15118 1/20 0.76
CASP3 P42574 1/20 0.76
SENP8 Q96LD8 1/20 0.76
SENP7 Q9BQF6 1/20 0.76
SENP6 Q9GZR1 1/20 0.76
TDP1 Q9NUW8 2/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
MEN1 O00255 1/20 0.59
GAA P10253 1/20 0.59
KMT2A Q03164 1/20 0.59
ALDH1A1 P00352 2/20 0.56
HPGD P15428 2/20 0.56
LMNA P02545 1/20 0.56
POLB P06746 1/20 0.56
TSHR P16473 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9084215 1.00 CYP1A2 (0.88) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL17266522 0.98 CYP1A2 (0.90) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL10458108 0.93 CYP1A2 (1.00) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL13698952 0.88 CYP1A2 (0.68) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL5708657 0.88 CYP1A2 (0.68) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL10421957 0.86 RAB9A (1.00) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL8621890 0.86 CYP1A2 (0.70) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL8918661 0.84 CYP1A2 (0.62) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL8617387 0.83 CYP1A2 (0.65) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2
SCHEMBL9081746 0.83 CYP1A2 (0.65) CYP1A2CYP2D6CYP2C19RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624917-A Method of inhibiting squalene synthetase TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-29 US disclosed
EP-0541037-A2 Squalene synthetase inhibitory composition and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-05-12 EP disclosed