SCHEMBL8915825

SCHEMBL8915825

O=C1c2ccccc2C(=O)N1CCCCCCCSc1ncccn1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.63
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C19 P33261 1/20 0.57
ALDH1A1 P00352 2/20 0.54
HPGD P15428 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
HSD17B10 Q99714 2/20 0.54
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
TSHR P16473 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HTR1A P08908 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
KDM1A O60341 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915123 1.00 MAPK1 (0.63) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8915242 1.00 MAPK1 (0.63) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8915923 1.00 MAPK1 (0.63) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL11315099 0.94 MAPK1 (0.67) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL9084403 0.88 MAPK1 (0.71) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL10679952 0.87 MAPK1 (0.51) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8618060 0.84 HSD17B10 (0.56) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL10674136 0.82 CYP1A2 (0.55) MAPK1CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8914866 0.80 CYP1A2 (0.88) CYP1A2CYP2D6CYP2C19ALDH1A1HPGD
SCHEMBL9084215 0.80 CYP1A2 (0.88) CYP1A2CYP2D6CYP2C19ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624917-A Method of inhibiting squalene synthetase TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-29 US disclosed
EP-0541037-A2 Squalene synthetase inhibitory composition and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-05-12 EP disclosed