SCHEMBL8916902

SCHEMBL8916902

N#CN=C(NCCCCCCOc1cccc(Cl)c1)Nc1ccncc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.64
NAMPT P43490 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
NOTUM Q6P988 2/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.39
F2 P00734 2/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
GALR3 O60755 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HRH3 Q9Y5N1 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918236 0.89 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL810990 0.89 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8917545 0.89 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL16312347 0.89 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL12083293 0.89 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL7142976 0.88 IKBKB (0.79) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL7148798 0.88 IKBKB (0.79) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL14212484 0.86 IKBKB (0.52) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL3825375 0.85 IKBKB (0.58) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8918926 0.85 IKBKB (0.61) IKBKBNAMPTCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696140-A FOR TREATMENT OF ASTHMA, ALLERGIES, NERVOUS SYSTEM DISORDERS OR CANCER LEO PHARMACEUTICAL PRODUCTS LTD. (DK) 1997-12-09 US disclosed