SCHEMBL8917353

SCHEMBL8917353

Fc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(S)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.68
PTGS1 P23219 11/20 0.68
CYP2C9 P11712 3/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
TSHR P16473 1/20 0.54
CYP2C19 P33261 1/20 0.54
THPO P40225 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
HIF1A Q16665 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6263143 0.87 PTGS2 (0.70) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5694394 0.87 PTGS2 (0.86) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL6266521 0.87 PTGS1 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL6610915 0.87 PTGS1 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL18448102 0.86 PTGS2 (0.72) PTGS2PTGS1CYP2C9CYP3A4TSHR
SCHEMBL8265772 0.86 PTGS2 (0.73) PTGS2PTGS1CYP2C9CYP3A4TSHR
SCHEMBL4587051 0.86 PTGS2 (0.73) PTGS2PTGS1CYP2C9CYP3A4TSHR
SCHEMBL27602805 0.85 PTGS1 (0.82) PTGS2PTGS1
SCHEMBL6266112 0.84 PTGS2 (0.87) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL6696373 0.84 PTGS2 (0.59) PTGS2PTGS1CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO disclosed