SCHEMBL8917471

SCHEMBL8917471

O=C(/C=C\c1[nH]cnc1-c1ccccc1)NC(Cc1ccccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
HTT P42858 2/20 0.44
NCOA1 Q15788 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
GSK3B P49841 2/20 0.43
QPCT Q16769 1/20 0.42
TACR3 P29371 1/20 0.42
CCR3 P51677 1/20 0.40
NOS2 P35228 1/20 0.39
FLT1 P17948 1/20 0.39
KDR P35968 1/20 0.39
TEK Q02763 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SOAT1 P35610 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912165 1.00 ALDH1A1 (0.44) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL8912159 0.76 ALDH1A1 (0.44) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL8913214 0.75 FLT1 (0.51) ALDH1A1HTTSMN1; SMN2FLT1KDR
Hydrochloric Acid SCHEMBL8914887 0.74 FLT1 (0.50) ALDH1A1HTTSMN1; SMN2FLT1KDR
Hydrochloric Acid SCHEMBL8913289 0.74 FLT1 (0.50) ALDH1A1HTTSMN1; SMN2FLT1KDR
SCHEMBL24157992 0.71 ALDH1A1 (0.58) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL28202339 0.70 ALDH1A1 (0.60) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL8912900 0.68 ALDH1A1 (0.42) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL8912912 0.68 ALDH1A1 (0.42) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL9716965 0.68 CNR2 (0.49) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5606073-A INTERMEDIATES FOR ADENOSINE ANTAGONISTS EISAI CO., LTD. (JP) 1997-02-25 US disclosed
US-5541213-A ADENOSINE A1 RECEPTOR ANTAGONISTS, TREATMENT OF KIDNEY DISORDERS EISAI CO., LTD. (JP) 1996-07-30 US disclosed
EP-0630894-A1 Propenoic acid derivatives as adenosine A1 antagonists Eisai Co., Ltd. (JP) 1994-12-28 EP disclosed