SCHEMBL8917576

SCHEMBL8917576

O=C(CF)Nc1cccnc1N1CCNCC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
MAPK1 P28482 1/20 0.45
CHEK1 O14757 1/20 0.44
POLB P06746 2/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
GAA P10253 1/20 0.44
HTR2C P28335 2/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR1A P08908 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22597906 0.83 EPHX2 (0.49) EPHX2MAPK1CHEK1ALDH1A1TSHR
SCHEMBL8918450 0.82 EPHX2 (0.56) EPHX2MAPK1CHEK1GAAHTR2C
SCHEMBL9376237 0.78 EPHX2 (0.48) EPHX2MAPK1CHEK1HTR2CHTR3E
SCHEMBL8919131 0.77 EPHX2 (0.52) EPHX2ALDH1A1HTR2CHTR3EHTR3B
SCHEMBL8923780 0.76 HDAC1 (0.52) MAPK1
Propionic Acid SCHEMBL9640910 0.75 PARP1 (0.53) EPHX2ALDH1A1HTR2CHTR3EHTR3B
SCHEMBL9036740 0.75 EPHX2 (0.55) EPHX2ALDH1A1HTR2CHTR3EHTR3B
SCHEMBL8916125 0.75 EPHX2 (0.59) EPHX2ALDH1A1HTR2CHTR3EHTR3B
SCHEMBL3334093 0.74 EPHX2 (0.51) EPHX2HTR2CHTR3EHTR3BHTR1A
Hydrochloric Acid SCHEMBL8703350 0.73 EPHX2 (0.50) EPHX2ALDH1A1HTR2CHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
US-5563142-A INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1996-10-08 US disclosed
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP disclosed
US-5489593-A Anti-aids piperazines THE UPJOHN COMPANY (US) 1996-02-06 US disclosed
EP-0594702-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS. UPJOHN CO (US) 1994-05-04 EP disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed