SCHEMBL9376237

SCHEMBL9376237

FC(F)(F)CNc1cccnc1N1CCNCC1.O=C(Nc1cccnc1N1CCNCC1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
HRH4 Q9H3N8 2/20 0.41
CHEK1 O14757 1/20 0.40
PRKCA P17252 1/20 0.40
FLT3 P36888 1/20 0.40
GSK3B P49841 1/20 0.40
PRKCQ Q04759 1/20 0.40
MAPK1 P28482 1/20 0.40
SCN9A Q15858 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
METAP2 P50579 1/20 0.39
PARP1 P09874 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2C P28335 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918450 0.92 EPHX2 (0.56) EPHX2CHEK1PRKCAFLT3GSK3B
SCHEMBL8916125 0.89 EPHX2 (0.59) EPHX2HRH4METAP2HTR3EHTR3B
SCHEMBL9375677 0.79 SLC29A1 (0.51) EPHX2
SCHEMBL8917576 0.78 EPHX2 (0.49) EPHX2CHEK1MAPK1HTR3EHTR3B
SCHEMBL22597906 0.76 EPHX2 (0.49) EPHX2CHEK1MAPK1HTR3EHTR3B
SCHEMBL8919131 0.74 EPHX2 (0.52) EPHX2FLT3HTR3EHTR3BHTR1A
Propionic Acid SCHEMBL9640910 0.74 PARP1 (0.53) EPHX2PARP1HTR3EHTR3BHTR1A
SCHEMBL3334093 0.73 EPHX2 (0.51) EPHX2FLT3PARP1HTR3EHTR3B
SCHEMBL7833448 0.72 CHEK1 (0.50) CHEK1MAPK1
Hydrochloric Acid SCHEMBL8703350 0.72 EPHX2 (0.50) EPHX2FLT3PARP1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0594702-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS. UPJOHN CO (US) 1994-05-04 EP disclosed