SCHEMBL8917883

SCHEMBL8917883

CCCNc1cccnc1N1CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
FLT3 P36888 1/20 0.47
TYRO3 Q06418 1/20 0.47
MERTK Q12866 1/20 0.47
GAS6 Q14393 1/20 0.47
HTR2C P28335 2/20 0.45
HRH4 Q9H3N8 1/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR1A P08908 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
KHK P50053 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3334093 0.89 EPHX2 (0.51) EPHX2FLT3TYRO3MERTKGAS6
Water SCHEMBL8415043 0.87 EPHX2 (0.50) EPHX2FLT3TYRO3MERTKGAS6
Hydrochloric Acid SCHEMBL8703350 0.87 EPHX2 (0.50) EPHX2FLT3TYRO3MERTKGAS6
Hydrochloric Acid SCHEMBL9076651 0.86 PARP1 (0.49) EPHX2FLT3TYRO3MERTKGAS6
SCHEMBL8919131 0.86 EPHX2 (0.52) EPHX2FLT3TYRO3MERTKGAS6
SCHEMBL8699158 0.82 EPHX2 (0.51) EPHX2HTR2CHTR3EHTR3BHTR1A
SCHEMBL9036740 0.81 EPHX2 (0.55) EPHX2HTR2CHTR3EHTR3BHTR1A
Propionic Acid SCHEMBL9640910 0.81 PARP1 (0.53) EPHX2HTR2CHTR3EHTR3BHTR1A
SCHEMBL8916125 0.81 EPHX2 (0.59) EPHX2HTR2CHRH4HTR3EHTR3B
SCHEMBL7868168 0.80 EPHX2 (0.48) EPHX2HTR2CHTR3EHTR3BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
EP-0594702-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS. UPJOHN CO (US) 1994-05-04 EP disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed