SCHEMBL8917936

SCHEMBL8917936

CC(=O)N1CCc2c(sc(C)c2CCN2CCC(c3noc4ccc(F)cc34)CC2)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.53
DRD3 P35462 3/20 0.53
HTR7 P34969 3/20 0.50
HTT P42858 1/20 0.49
DRD2 P14416 2/20 0.47
KCNH2 Q12809 2/20 0.47
ALDH1A1 P00352 1/20 0.47
SLC22A2 O15244 1/20 0.47
CACNA1F O60840 1/20 0.47
ADRB2 P07550 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
HTR1A P08908 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2A P08913 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
TSHR P16473 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916147 0.94 DRD2 (0.54) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8916687 0.89 DRD2 (0.54) HTR2ADRD3DRD2KCNH2CHRM2
SCHEMBL8917929 0.88 DRD2 (0.54) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8920271 0.87 DRD2 (0.56) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8916567 0.86 DRD2 (0.55) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8918134 0.86 DRD2 (0.53) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8916465 0.85 HTR2A (0.53) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8918706 0.85 DRD2 (0.56) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8918054 0.85 DRD2 (0.54) HTR2ADRD3HTR7DRD2KCNH2
SCHEMBL8916981 0.84 HTR2A (0.53) HTR2ADRD3HTR7DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed