SCHEMBL8918692

SCHEMBL8918692

O=C(O)NC(Cc1ccc2ccccc2c1)C(O)CCl

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.46
MME P08473 5/20 0.44
ACE P12821 4/20 0.44
CPA1 P15085 2/20 0.44
ACE2 Q9BYF1 2/20 0.44
FCER2 P06734 2/20 0.43
MMP9 P14780 2/20 0.43
MMP8 P22894 2/20 0.43
CCR1 P32246 1/20 0.43
CA2 P00918 1/20 0.42
CYP1A2 P05177 1/20 0.41
CTSD P07339 2/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918697 1.00 TACR1 (0.46) TACR1MMEACECPA1ACE2
SCHEMBL8919979 0.85 MME (0.47) TACR1MMEACECPA1ACE2
SCHEMBL6944317 0.84 BACE1 (0.47) CYP1A2
SCHEMBL2712694 0.84 BACE1 (0.47) CYP1A2
SCHEMBL10707926 0.84 BACE1 (0.47) CYP1A2
SCHEMBL2712697 0.84 BACE1 (0.47) CYP1A2
SCHEMBL6944939 0.84 BACE1 (0.47) CYP1A2
SCHEMBL6944942 0.84 BACE1 (0.47) CYP1A2
SCHEMBL8919984 0.83 MME (0.44) TACR1MMEACECPA1ACE2
SCHEMBL12805325 0.80 MME (0.51) TACR1MMEACECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed