SCHEMBL8919984

SCHEMBL8919984

C[C@H](O)CC(CCl)[C@H](Cc1ccc2ccccc2c1)NC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MME P08473 6/20 0.44
ACE P12821 5/20 0.44
CPA1 P15085 2/20 0.44
ACE2 Q9BYF1 2/20 0.44
MMP9 P14780 5/20 0.43
MMP8 P22894 5/20 0.43
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
TACR1 P25103 1/20 0.41
CCR1 P32246 1/20 0.41
PSMB5 P28074 3/20 0.41
FCER2 P06734 1/20 0.41
PSMB1 P20618 1/20 0.40
PSMB2 P49721 1/20 0.40
MMP2 P08253 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918697 0.83 TACR1 (0.46) MMEACECPA1ACE2MMP9
SCHEMBL8918692 0.83 TACR1 (0.46) MMEACECPA1ACE2MMP9
SCHEMBL8919979 0.79 MME (0.47) MMEACECPA1ACE2MMP9
SCHEMBL8919990 0.78 HTR2A (0.46) MMEACECPA1ACE2MMP9
SCHEMBL12805325 0.77 MME (0.51) MMEACECPA1ACE2MMP9
SCHEMBL7291159 0.76 HTR2A (0.44) MMEACECPA1ACE2MMP9
SCHEMBL8921872 0.71 CTSG (0.52) MMEACECPA1ACE2MMP9
SCHEMBL8921880 0.71 CTSG (0.52) MMEACECPA1ACE2MMP9
SCHEMBL8919989 0.71 PIN1 (0.41) MMEACECPA1ACE2MMP9
SCHEMBL7436981 0.70 TACR1 (0.51) MMEACECPA1ACE2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed