SCHEMBL8918941

SCHEMBL8918941

N#CN=C(NCCSc1ccccc1)Nc1cncc(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
ALDH1A1 P00352 3/20 0.54
HRH4 Q9H3N8 8/20 0.42
HRH2 P25021 7/20 0.42
HRH1 P35367 5/20 0.41
HRH3 Q9Y5N1 5/20 0.41
CASP3 P42574 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
RECQL P46063 1/20 0.36
HDAC4 P56524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915168 0.82 NPC1 (0.50) NPC1RAB9ASMN1; SMN2ALDH1A1HRH4
SCHEMBL7430606 0.82 POLB (0.53) SMN1; SMN2HRH4HRH2HRH1CASP3
SCHEMBL8921944 0.81 NPC1 (0.46) NPC1RAB9ASMN1; SMN2ALDH1A1HRH4
SCHEMBL8918934 0.79 HRH4 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1HRH4
SCHEMBL8918937 0.79 HRH4 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1HRH4
SCHEMBL7359985 0.73 KCNJ11 (0.40) ALDH1A1HDAC4MAPTHTT
SCHEMBL7359989 0.73 KCNJ11 (0.40) ALDH1A1HDAC4MAPTHTT
SCHEMBL7359997 0.73 KCNJ11 (0.40) ALDH1A1HDAC4MAPTHTT
SCHEMBL3408797 0.70 SMN1; SMN2 (1.00) NPC1RAB9ASMN1; SMN2ALDH1A1CASP3
SCHEMBL29858769 0.70 SMN1; SMN2 (1.00) NPC1RAB9ASMN1; SMN2ALDH1A1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696140-A FOR TREATMENT OF ASTHMA, ALLERGIES, NERVOUS SYSTEM DISORDERS OR CANCER LEO PHARMACEUTICAL PRODUCTS LTD. (DK) 1997-12-09 US disclosed
US-5563160-A NERVOUS SYSTEM DISORDERS, ANTIHISTAMINE, ANTIALLERGENS Leo Pharmaceutical Products Ltd. A/S (L.o slashed.vens Kemiske Fabrik Produktionsaktieselskab) (DK) 1996-10-08 US disclosed
EP-0660823-B1 N-CYANO-N'-PYRIDYLGUANIDINES AS SEROTONIN ANTAGONISTS LEO PHARM PROD LTD (DK) 1996-08-14 EP disclosed