SCHEMBL8919916

SCHEMBL8919916

O=c1[nH]c2cc(Cl)ccc2c(O)c1OCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.53
POLB P06746 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
BLM P54132 1/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRIN2B Q13224 1/20 0.50
GRIN2C Q14957 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8783837 0.82 CYP1A2 (0.74) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL8783655 0.80 CYP1A2 (0.75) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL16632110 0.78 HDAC1 (0.46) TSHRMEN1KMT2AALDH1A1MAPT
SCHEMBL8920123 0.75 KDM4E (0.52) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL8920155 0.74 KDM4E (0.54) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL1612505 0.73 KDM4E (0.79) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL8921277 0.73 MEN1 (0.49) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL27486624 0.72 CYP1A2 (0.50) CYP1A2POLBCYP3A4CYP2C9TSHR
SCHEMBL8784817 0.72 KDM4E (0.69) CYP1A2MEN1KMT2AKDM4ECYP2D6
SCHEMBL7121201 0.71 ALDH1A1 (0.53) TSHRMEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US claimed
CN-1120538-A 3-heteroaliphatyl- and 3-hetero (aryl) aliphatyl-2(1H)-quinolone dericatives CIBA GEIGY AG (CH) 1996-04-17 CN claimed