SCHEMBL8920189

SCHEMBL8920189

O/N=C1\CCC(c2ccc(F)cc2)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP19A1 P11511 1/20 0.38
PRCP P42785 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
HTR2A P28223 4/20 0.36
HTR2C P28335 4/20 0.36
HTR2B P41595 4/20 0.36
HRH3 Q9Y5N1 4/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920191 1.00 HPGD (0.38) HPGDL3MBTL1CYP19A1PRCPNPSR1
SCHEMBL4867731 0.85 CYP3A4 (0.40)
SCHEMBL8924522 0.85 HPGD (0.38) HPGDL3MBTL1CYP19A1PRCPNPSR1
SCHEMBL8921189 0.85 HTT (0.40) HPGDL3MBTL1
SCHEMBL8921192 0.85 HTT (0.40) HPGDL3MBTL1
SCHEMBL4867739 0.85 CYP3A4 (0.40)
SCHEMBL8924511 0.85 HPGD (0.38) HPGDL3MBTL1CYP19A1PRCPNPSR1
SCHEMBL8920936 0.82 HPGD (0.40) HPGDL3MBTL1CYP19A1NPSR1SMN1; SMN2
SCHEMBL8920925 0.82 HPGD (0.40) HPGDL3MBTL1CYP19A1NPSR1SMN1; SMN2
SCHEMBL10041960 0.79 SLC6A2 (0.51) HTR2AHTR2CHTR2BHRH3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed