SCHEMBL8921189

SCHEMBL8921189

O/N=C1\CCC(c2ccc(Cl)cc2)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921192 1.00 HTT (0.40) HTTHPGDL3MBTL1SLC6A2SLC6A4
SCHEMBL8920189 0.85 HPGD (0.38) HPGDL3MBTL1
SCHEMBL8924511 0.85 HPGD (0.38) HPGDL3MBTL1SLC6A2SLC6A4SLC6A3
SCHEMBL8920191 0.85 HPGD (0.38) HPGDL3MBTL1
SCHEMBL8924522 0.85 HPGD (0.38) HPGDL3MBTL1SLC6A2SLC6A4SLC6A3
SCHEMBL10041960 0.85 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3
SCHEMBL8920192 0.85 HTT (0.40) HTTHPGDL3MBTL1
SCHEMBL10041954 0.85 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3
SCHEMBL20436754 0.85 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3
SCHEMBL8920198 0.85 HTT (0.40) HTTHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed