SCHEMBL8920561

SCHEMBL8920561

NC(=O)CN1C(=O)C(Br)CC(c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 14/20 0.49
FDFT1 P37268 1/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP2C19 P33261 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542926 0.89 CCKBR (0.49) CCKBRFDFT1MEN1KMT2ACYP2C19
SCHEMBL8921634 0.87 CCKBR (0.47) CCKBRMEN1KMT2ACYP2C19
SCHEMBL8923711 0.87 CCKBR (0.47) CCKBRCYP2C19
SCHEMBL9366810 0.86 CYP2C19 (0.47) CCKBRKMT2ACYP2C19
SCHEMBL8920295 0.86 CCKBR (0.51) CCKBRKMT2ACYP2C19
SCHEMBL8401370 0.80 CCKBR (0.48) CCKBR
SCHEMBL8922239 0.80 SLC6A2 (0.42) CYP2C19
SCHEMBL9541588 0.79 CCKBR (0.78) CCKBR
SCHEMBL8399132 0.79 CCKBR (0.50) CCKBRCYP2C19
SCHEMBL8922081 0.78 CYP2C19 (0.43) CCKBRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed