SCHEMBL8921056

SCHEMBL8921056

O=C1CCC(c2ccccc2)CC1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.46
CRBN Q96SW2 1/20 0.46
SRD5A1 P18405 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C1 Q04828 1/20 0.40
HSD11B1 P28845 2/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CYP19A1 P11511 1/20 0.38
MAOB P27338 1/20 0.38
SLC18A3 Q16572 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29016897 0.81 DDB1 (0.61) DDB1CRBNHSD11B1CYP19A1MAOB
SCHEMBL31147295 0.79 SRD5A1 (0.43) SRD5A1AKR1C3AKR1C1
SCHEMBL8676176 0.79 MT-CO2 (0.49) DDB1CRBNHSD11B1ALDH1A1CYP19A1
SCHEMBL5845789 0.79 DDB1 (0.47) DDB1CRBNHSD11B1CYP19A1MAOB
SCHEMBL7739386 0.79 SRD5A1 (0.38) SRD5A1AKR1C3AKR1C1ALDH1A1SLC18A3
SCHEMBL11701944 0.77 KDM4E (0.46) SRD5A1AKR1C3AKR1C1ALDH1A1POLB
SCHEMBL11777020 0.76 DDB1 (0.45) DDB1CRBNHSD11B1CYP19A1MAOB
SCHEMBL22321333 0.76 SRD5A1 (0.45) DDB1CRBNSRD5A1AKR1C3AKR1C1
SCHEMBL13039616 0.75 SRD5A1 (0.47) SRD5A1AKR1C3AKR1C1HPGDMAOB
SCHEMBL28391454 0.75 DDB1 (0.44) DDB1CRBNHSD11B1TSHRCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107338043-B Novel racemic chiral organic boron-nitrogen fluorescent compound and preparation method thereof 湖南大学 2020-04-24 CN disclosed
CN-107338043-A A kind of new racemic chirality organic boron nitrogen fluorescent chemicals and preparation method thereof 湖南大学 2017-11-10 CN disclosed
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed