SCHEMBL8921064

SCHEMBL8921064

C=CC(Cn1c(N)nc2nc[nH]c2c1=O)OCP(=O)(O)O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 5/20 0.35
ADORA2A P29274 4/20 0.35
CDK1 P06493 4/20 0.34
CCNB1 P14635 4/20 0.34
CCNA2 P20248 4/20 0.34
CDK2 P24941 4/20 0.34
CCNA1 P78396 4/20 0.34
MGMT P16455 3/20 0.34
HPRT1 P00492 2/20 0.33
FGFR1 P11362 1/20 0.33
SLC22A6 Q4U2R8 1/20 0.32
PDE4A P27815 3/20 0.32
PDE4B Q07343 3/20 0.32
PDE4C Q08493 3/20 0.32
PDE4D Q08499 3/20 0.32
ADORA3 P0DMS8 1/20 0.32
CFTR P13569 1/20 0.32
PNP P00491 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170817 0.84 HPRT1 (0.43) ADORA2BADORA2ACDK1CCNB1CCNA2
SCHEMBL16020626 0.82 HPRT1 (0.43) ADORA2BADORA2AMGMTHPRT1FGFR1
SCHEMBL8918790 0.82 ADORA2B (0.37) ADORA2BADORA2ACDK1CCNB1CCNA2
SCHEMBL216787 0.76 HPRT1 (0.44) ADORA2BADORA2AHPRT1FGFR1SLC22A6
SCHEMBL6836084 0.76 HPRT1 (0.35) ADORA2BADORA2ACDK1CCNB1CCNA2
SCHEMBL385154 0.75 CDK1 (0.38) ADORA2BCDK1CCNB1CCNA2CDK2
SCHEMBL16037341 0.74 CDK1 (0.40) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL2249888 0.74 ADORA2A (0.39) ADORA2BADORA2ACDK1CCNB1CCNA2
SCHEMBL15545146 0.74 HPRT1 (0.42) ADORA2BADORA2ACDK1CCNB1CCNA2
SCHEMBL669007 0.73 ADORA2B (0.61) ADORA2BADORA2ACDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696263-A Antiviral acyclic phosphonomethoxyalkylsubstituted alkenyl and alkynyl purine and pyrimidine derivatives INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1997-12-09 US claimed
US-5696263-A Antiviral acyclic phosphonomethoxyalkylsubstituted alkenyl and alkynyl purine and pyrimidine derivatives INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1997-12-09 US disclosed