SCHEMBL8922074

SCHEMBL8922074

O=C(CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1(c2ccccc2)CCNCC1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.67
SLC6A4 P31645 8/20 0.52
KCNH2 Q12809 1/20 0.45
OPRM1 P35372 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8924174 0.99 TACR1 (0.65) TACR1SLC6A4KCNH2OPRM1
Hydrochloric Acid SCHEMBL8114977 0.87 TACR1 (0.68) TACR1SLC6A4KCNH2OPRM1
SCHEMBL6485653 0.74 TACR1 (0.74) TACR1KCNH2
SCHEMBL6485655 0.74 TACR1 (0.74) TACR1KCNH2
SCHEMBL8920152 0.74 TACR1 (1.00) TACR1SLC6A4KCNH2
SCHEMBL8922535 0.74 TACR1 (0.59) TACR1SLC6A4KCNH2
SCHEMBL4261726 0.74 OPRM1 (0.62) TACR1SLC6A4KCNH2OPRM1
Hydrochloric Acid SCHEMBL8924192 0.73 TACR1 (0.97) TACR1SLC6A4KCNH2
Hydrochloric Acid SCHEMBL8919189 0.73 TACR1 (0.58) TACR1SLC6A4KCNH2
Hydrochloric Acid SCHEMBL1308247 0.72 OPRM1 (0.61) TACR1SLC6A4KCNH2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995004042-A1 4-PHENYL-4-PHENYLPROPYL(ENYL)-PIPERIDINES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-02-09 WO claimed
US-5663352-A 4-phenyl-4-phenylpropyl(enyl)-piperidines as tachykinin antagonists MERCK SHARP & DOHME LIMITED (GB) 1997-09-02 US disclosed
EP-0711281-A1 4-PHENYL-4-PHENYLPROPYL(ENYL)-PIPERIDINES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1996-05-15 EP disclosed
WO-1995004042-A1 4-PHENYL-4-PHENYLPROPYL(ENYL)-PIPERIDINES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-02-09 WO disclosed