SCHEMBL8924144

SCHEMBL8924144

CC(Br)c1cc2nc(NC(=O)C(C)(C)C)[nH]c(=O)c2c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 2/20 0.39
TYMS P04818 4/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 1/20 0.38
XBP1 P17861 1/20 0.38
POLB P06746 2/20 0.37
TSHR P16473 1/20 0.37
ADORA1 P30542 1/20 0.37
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651272 0.84 TYMS (0.47) RAB9ANPC1MEN1KMT2ACYP1A2
SCHEMBL6649736 0.83 TYMS (0.56) RAB9ANPC1MEN1KMT2ACYP1A2
SCHEMBL8924156 0.82 TYMS (0.46) RAB9ANPC1MEN1KMT2ACYP1A2
SCHEMBL6650303 0.77 TYMS (0.58) RAB9ANPC1MEN1KMT2ACYP1A2
SCHEMBL6650779 0.73 TYMS (0.62) SMN1; SMN2ALDH1A1HPGDTYMSMAPT
SCHEMBL1369022 0.72 ALDH1A1 (0.45) RAB9ANPC1MEN1KMT2ACYP1A2
SCHEMBL6447534 0.72 TYMS (0.56) SMN1; SMN2ALDH1A1KDM4EHPGDTYMS
SCHEMBL6652207 0.71 TYMS (0.57) SMN1; SMN2ALDH1A1HPGDTYMS
SCHEMBL6455693 0.71 TYMS (0.46) SMN1; SMN2ALDH1A1HPGDTYMSMAPT
SCHEMBL6649923 0.70 TYMS (0.59) RAB9ANPC1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661155-A THYMIDYLATE SYNTHASE INHIBITOR; ADMINISTERING TO THE MAMMAL SUFFERING FROM LEUKEMIA OR TUMOR 2-(5-(((1,2-DIHYDRO-3-METHYL-1-OXOBENZO(F)QUINAZOLINE-9-YL) METHYL)AMINO)-1-OXO-2-ISOINDOLINYL)GLUTARIC ACID OR SALTS GLAXO WELLCOME INC. (US) 1997-08-26 US disclosed