SCHEMBL8924809

SCHEMBL8924809

O=C(CBr)c1cccc(-n2cncn2)n1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.39
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 3/20 0.34
POLB P06746 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GRK6 P43250 1/20 0.34
PTPN1 P18031 1/20 0.33
CYP2A6 P11509 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
STING1 Q86WV6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18168008 0.82 KDM4E (0.50) IRAK4ALDH1A1MAPTKDM4EPOLB
SCHEMBL28303005 0.76 CYP2A6 (0.47) ALDH1A1MAPTKDM4EPOLBMEN1
SCHEMBL28712036 0.74 KDM4E (0.52) KDM4EPOLBKMT2APTPN1
SCHEMBL5769923 0.72 CYP2A6 (0.41) ALDH1A1MAPTKDM4EPOLBMEN1
SCHEMBL14376686 0.71 MAPT (0.58) ALDH1A1MAPTKDM4EPOLBMEN1
SCHEMBL16419707 0.71 IRAK4 (0.38) IRAK4ALDH1A1MAPTKDM4EPOLB
SCHEMBL20187481 0.70 MAPT (0.34) ALDH1A1MAPTKDM4EPOLBMEN1
SCHEMBL20209382 0.69 MAPT (0.33) MAPTKDM4EPOLBHTTSMN1; SMN2
SCHEMBL8923789 0.69 HSD17B14 (0.53) ALDH1A1KDM4E
SCHEMBL8925427 0.69 GSK3B (0.52) IRAK4ALDH1A1KDM4EKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639770-A SUPEROXIDE INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-06-17 US disclosed
EP-0600092-A1 THIAZOLE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-08 EP disclosed