SCHEMBL8925686

SCHEMBL8925686

CCOC(=O)/C(=C/NC1CC1)C(=O)c1c(C(F)(F)F)cc(F)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.38
EPHX2 P34913 1/20 0.37
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 2/20 0.35
POLB P06746 2/20 0.35
LMNA P02545 2/20 0.34
MAPK1 P28482 1/20 0.34
MAPT P10636 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 3/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
DHODH Q02127 2/20 0.32
GPR35 Q9HC97 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8925690 1.00 NPSR1 (0.38) NPSR1EPHX2ALDH1A1L3MBTL1KDM4E
SCHEMBL9501196 0.88 NPSR1 (0.36) NPSR1ALDH1A1POLBLMNAMAPT
SCHEMBL1348749 0.86 POLB (0.39) NPSR1ALDH1A1KDM4EPOLBLMNA
SCHEMBL1348752 0.86 POLB (0.39) NPSR1ALDH1A1KDM4EPOLBLMNA
SCHEMBL8733953 0.84 NPSR1 (0.39) NPSR1EPHX2ALDH1A1KDM4EPOLB
SCHEMBL8733952 0.84 NPSR1 (0.39) NPSR1EPHX2ALDH1A1KDM4EPOLB
SCHEMBL1345391 0.83 CYP2D6 (0.38) NPSR1ALDH1A1LMNAMAPK1MAPT
SCHEMBL9562436 0.83 CYP2D6 (0.38) NPSR1ALDH1A1LMNAMAPK1MAPT
SCHEMBL1345392 0.83 CYP2D6 (0.38) NPSR1ALDH1A1LMNAMAPK1MAPT
SCHEMBL5505218 0.83 POLB (0.37) NPSR1ALDH1A1KDM4EPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648567-A INTERMEDIATES FOR BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-07-15 US disclosed
US-5493048-A REACTING METALLIZED FLUORO-TRIFLUOROMETHYLBENZENE DERIVATIVE WITH CARBON DIOXIDE AND PRODUCT IS THEN HYDROLYSED WITH AN ACID TO FORM ACID, SIMILARLY HALOGENATION GIVE ACID HALIDE AND WITH ALCOHOL GIVES ESTER BAYER AKTIENGESELLSCHAFT (DE) 1996-02-20 US disclosed
US-5457104-A Antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1995-10-10 US disclosed