SCHEMBL8926434

SCHEMBL8926434

Clc1cccc(OC[C@@H]2CNCCO2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.53
SLC6A4 P31645 4/20 0.53
SLC6A2 P23975 2/20 0.53
HTR2B P41595 2/20 0.53
SLC6A3 Q01959 2/20 0.53
ADRB2 P07550 1/20 0.53
HTR1A P08908 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA2C P18825 1/20 0.53
HRH1 P35367 1/20 0.50
OPRD1 P41143 1/20 0.50
OPRK1 P41145 1/20 0.50
HTR3A P46098 1/20 0.50
EPHA2 P29317 2/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HIF1A Q16665 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3162540 1.00 HTR2A (0.53) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL31381402 0.90 CYP3A4 (0.60) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL26668483 0.90 CYP3A4 (0.60) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL26668476 0.90 CYP3A4 (0.60) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL1698274 0.84 ADRA2C (0.64) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL17277433 0.84 SLC6A4 (0.56) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL21254308 0.84 SLC6A4 (0.53) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL9814604 0.84 SLC6A4 (0.53) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL8926009 0.83 HTR2A (0.55) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL8926000 0.83 HTR2A (0.55) HTR2ASLC6A4SLC6A2HTR2BSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614518-A Morpholine derivatives as dopamine receptor subtype ligands MERCK SHARP & DOHME LTD. (GB) 1997-03-25 US disclosed