SCHEMBL8927622

SCHEMBL8927622

CC(=O)NCCN(C)CCN

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PAOX Q6QHF9 3/20 0.50
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
HIF1A Q16665 1/20 0.43
MTNR1A P48039 9/20 0.42
MTNR1B P49286 9/20 0.42
TSHR P16473 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADRA1A P35348 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13407441 0.89 KDM4E (0.52) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL1583774 0.83 CARM1 (0.34) PAOXKDM4EMTNR1AMTNR1B
SCHEMBL15270870 0.81 PAOX (0.32) PAOXKDM4E
SCHEMBL9547380 0.81 KDM4E (0.44) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL17393151 0.81 KDM4E (0.44) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL20725629 0.81 PAOX (0.52) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL12265757 0.81 KDM4E (0.44) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL18506889 0.81 PAOX (0.45) PAOXKDM4EMAPK1HIF1AMTNR1A
SCHEMBL21017754 0.79 POLB (0.37) KDM4EALDH1A1
SCHEMBL15146684 0.78 KDM4E (0.46) PAOXKDM4EMAPK1HIF1AMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964617-B1 SUBSTITUTED BICYCLIC DIHYDROPYRIMIDINONES AND THEIR USE AS INHIBITORS OF NEUTROPHIL ELASTASE ACTIVITY BOEHRINGER INGELHEIM INT (DE) 2017-04-12 EP disclosed
US-5600025-A CHEMICAL INTERMEDIATES FOR NONWAXY FUEL AND LUBRICANT ADDITIVES CONTAINING ALKYLPHENYL POLY(OXYPROPYLENE) AMINOCARBAMATES; ANTIDEPOSIT AGENTS CHEVRON CHEMICAL COMPANY (US) 1997-02-04 US disclosed
EP-0419488-A4 LUBRICATING OIL COMPOSITIONS AND FUEL COMPOSITIONS CONTAINING SUBSTANTIALLY STRAIGHT CHAIN PINWHEEL ALKYLPHENYL POLY(OXYPROPYLENE) AMINOCARBAMATES CHEVRON RES (US) 1994-11-23 EP disclosed
US-5322529-A Liquid additive; internal combustion engines CHEVRON RESEARCH AND TECHNOLOGY COMPANY (US) 1994-06-21 US disclosed
EP-0419488-A1 LUBRICATING OIL COMPOSITIONS AND FUEL COMPOSITIONS CONTAINING SUBSTANTIALLY STRAIGHT CHAIN PINWHEEL ALKYLPHENYL POLY(OXYPROPYLENE) AMINOCARBAMATES CHEVRON U.S.A. Inc. (US) 1991-04-03 EP disclosed
WO-1990007564-A1 LUBRICATING OIL COMPOSITIONS AND FUEL COMPOSITIONS CONTAINING SUBSTANTIALLY STRAIGHT CHAIN PINWHEEL ALKYLPHENYL POLY(OXYPROPYLENE) AMINOCARBAMATES CHEVRON RESEARCH COMPANY (US) 1990-07-12 WO disclosed
US-4624681-A Dispersant additives for lubricating oils and fuels CHEVRON RESEARCH COMPANY (US) 1986-11-25 US disclosed
US-4198306-A HYDROCARBYL-POLY(OXYALKYLENE) AMINOESTERS, USED IN FUELS AND LUBRICATING OILS CHEVRON RESEARCH COMPANY (US) 1980-04-15 US disclosed