SCHEMBL8929641

SCHEMBL8929641

c1nc(Oc2ccc3c(c2)CCC3)c2cc[nH]c2n1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.62
TNNI3K Q59H18 2/20 0.53
JAK3 P52333 2/20 0.48
KDR P35968 5/20 0.44
BRAF P15056 1/20 0.43
MAPK14 Q16539 1/20 0.43
TTBK1 Q5TCY1 5/20 0.41
TTBK2 Q6IQ55 4/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830504 0.79 JAK2 (0.42) TRPA1JAK3
SCHEMBL4548928 0.78 KDR (0.74) TNNI3KKDRBRAFMAPK14MET
SCHEMBL8929278 0.77 TRPA1 (0.56) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL2882091 0.76 TRPA1 (0.75) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL30564544 0.76 TRPA1 (0.75) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL25793164 0.75 TRPA1 (0.80) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL29837326 0.75 TRPA1 (0.80) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL21593208 0.74 NR1H2 (0.56) TRPA1TNNI3KJAK3KDRBRAF
SCHEMBL7830506 0.74 PDPK1 (0.47) BRAF
SCHEMBL7821542 0.74 NPC1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed