SCHEMBL8931650

SCHEMBL8931650

CCC(C(=O)c1ccc(Cl)cc1)n1ncn(-c2ccc(N3CCN(c4cccc(OC)c4)CC3)nc2)c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.51
MAPT P10636 4/20 0.45
DRD4 P21917 8/20 0.44
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 3/20 0.40
DRD2 P14416 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
PMP22 Q01453 1/20 0.40
MAPK1 P28482 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CACNA1G O43497 1/20 0.39
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2C P18825 1/20 0.38
HRH2 P25021 1/20 0.38
HTR1B P28222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931730 0.92 MAPT (0.54) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8931682 0.91 DGAT1 (0.48) DGAT1MAPTDRD4ALDH1A1KDM4E
SCHEMBL8931698 0.91 DGAT1 (0.56) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8931744 0.90 DGAT1 (0.48) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8931641 0.90 DGAT1 (0.44) DGAT1MAPTDRD4CYP3A4DRD2
Hydrochloric Acid SCHEMBL8931711 0.89 DGAT1 (0.51) DGAT1MAPTDRD4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8931688 0.89 DGAT1 (0.47) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8927419 0.89 DGAT1 (0.47) DGAT1MAPTDRD4ALDH1A1KDM4E
SCHEMBL8931707 0.89 MAPT (0.54) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8931629 0.88 DGAT1 (0.51) DGAT1MAPTALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650411-A BACTERICIDES FOR HELICOBACTER DISEASES AND BACTERIA RESISTANCE JANSSEN PHARMACEUTICA N.V. (BE) 1997-07-22 US disclosed
EP-0684821-A1 SUBSTITUTED AZOLONE DERIVATIVES FOR TREATING DISEASES CAUSED BY HELICOBACTER JANSSEN PHARMACEUTICA N.V. (BE) 1995-12-06 EP disclosed
WO-1994018978-A1 SUBSTITUTED AZOLONE DERIVATIVES FOR TREATING DISEASES CAUSED BY HELICOBACTER JANSSEN PHARMACEUTICA N.V. (BE) 1994-09-01 WO disclosed