SCHEMBL8933318

SCHEMBL8933318

Cc1nc2sc3ccccc3c2c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.53
TYMS P04818 4/20 0.51
PARP1 P09874 5/20 0.50
ALDH1A1 P00352 4/20 0.50
TNKS2 Q9H2K2 3/20 0.50
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
NPC1 O15118 2/20 0.50
MAPT P10636 2/20 0.50
RAB9A P51151 2/20 0.50
ELANE P08246 1/20 0.47
CYP1A2 P05177 1/20 0.46
HIF1A Q16665 1/20 0.46
TNKS O95271 2/20 0.45
HPGD P15428 3/20 0.45
USP2 O75604 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30764972 0.83 TNKS (0.46) MAPK1TYMSALDH1A1TNKS2KDM4E
SCHEMBL6124884 0.81 TNKS2 (0.54) TYMSALDH1A1TNKS2KDM4EMAPT
SCHEMBL6124872 0.81 ELANE (0.44) MAPK1TYMSALDH1A1TNKS2KDM4E
SCHEMBL8198913 0.78 TNKS (0.42) TYMSALDH1A1TNKS2KDM4ESMN1; SMN2
SCHEMBL6124881 0.77 ELANE (0.44) MAPK1TYMSALDH1A1TNKS2KDM4E
SCHEMBL8191558 0.77 ALDH1A1 (0.62) MAPK1ALDH1A1KDM4ESMN1; SMN2MAPT
SCHEMBL7878783 0.74 ELANE (0.43) ALDH1A1TNKS2KDM4ESMN1; SMN2NPC1
SCHEMBL2689332 0.71 PDPK1 (0.50) PARP1ALDH1A1TNKS2SMN1; SMN2NPC1
SCHEMBL22988563 0.71 ELANE (0.43) ALDH1A1KDM4ESMN1; SMN2NPC1MAPT
SCHEMBL14043486 0.71 RXFP1 (0.40) MAPK1ALDH1A1TNKS2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022992-A1 TRICYCLIC SUBSTITUTED HEXAHYDROBENZ[E]ISOINDOLE ALPHA-1 ADRENERGIC ANTAGONISTS ABBOTT LABORATORIES (US) 1996-08-01 WO disclosed