SCHEMBL8933877

SCHEMBL8933877

NS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)c3c2-c2ccc(F)cc2CS3)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 1.00
PTGS1 P23219 12/20 1.00
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA3 P07451 1/20 0.51
CA4 P22748 1/20 0.51
CA6 P23280 1/20 0.51
CA5A P35218 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51
CA13 Q8N1Q1 1/20 0.51
CA14 Q9ULX7 1/20 0.51
CA5B Q9Y2D0 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698663 0.90 PTGS2 (0.82) PTGS2PTGS1
SCHEMBL8933971 0.89 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8933906 0.89 PTGS2 (0.80) PTGS2PTGS1CA12CA1CA2
SCHEMBL8933921 0.88 PTGS2 (1.00) PTGS2PTGS1CA12CA1CA2
SCHEMBL8933893 0.87 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8933896 0.84 PTGS2 (0.72) PTGS2PTGS1CA12CA1CA2
SCHEMBL8933829 0.84 PTGS2 (1.00) PTGS2PTGS1CA12CA1CA2
SCHEMBL8933812 0.83 PTGS2 (0.76) PTGS2PTGS1
SCHEMBL8933887 0.83 PTGS2 (0.71) PTGS2PTGS1CA12CA1CA2
SCHEMBL8933959 0.83 PTGS2 (0.71) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed