SCHEMBL8935897

SCHEMBL8935897

NC(COCc1ccccc1)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.70
CASP3 P42574 2/20 0.46
TACR1 P25103 3/20 0.45
LTA4H P09960 1/20 0.44
SLC1A1 P43005 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 2/20 0.41
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29811681 0.82 MAPK1 (1.00) MAPK1KMT2ATSHRRAB9AALDH1A1
SCHEMBL8935936 0.82 MAPK1 (1.00) MAPK1KMT2ATSHRRAB9AALDH1A1
SCHEMBL23144183 0.80 MAPK1 (0.67) MAPK1CASP3TDP1L3MBTL1KMT2A
SCHEMBL9575717 0.80 MAPK1 (0.67) MAPK1CASP3TDP1L3MBTL1KMT2A
SCHEMBL1529481 0.80 EPHX1 (0.53) MAPK1CASP3LTA4HTDP1L3MBTL1
SCHEMBL1529483 0.80 EPHX1 (0.53) MAPK1CASP3LTA4HTDP1L3MBTL1
SCHEMBL2370243 0.80 EPHX1 (0.53) MAPK1CASP3LTA4HTDP1L3MBTL1
SCHEMBL10052099 0.79 MAPK1 (0.65) MAPK1CASP3TDP1L3MBTL1KMT2A
SCHEMBL10949349 0.79 MAPK1 (0.57) MAPK1CASP3LTA4HSLC1A1TDP1
SCHEMBL10949350 0.79 MAPK1 (0.57) MAPK1CASP3TACR1SLC1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5531978-A CHELATE COMPOUNDS, IMAGING NYCOMED IMAGING AS (NO) 1996-07-02 US disclosed
US-5419893-A Aminopolycarboxylic acids and derivatives thereof for magnetic resonance imaging NYCOMED IMAGING AS (NO) 1995-05-30 US disclosed
US-5198208-A Chelate compounds for diagnosis by magnetic resonance imaging, ultrasound or radiation therapy NYCOMED IMAGING AS (NO) 1993-03-30 US disclosed
EP-0466200-A1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1992-01-15 EP disclosed
WO-1989000557-A1 AMINOPOLYCARBOXYLIC ACIDS AND DERIVATIVES THEREOF COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1989-01-26 WO disclosed